SCHEMBL14845241

SCHEMBL14845241

CCC(=C(C(=O)O)C(=O)c1ccc(F)c(F)c1F)N(C)C

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.50
CES1 P23141 3/20 0.50
BCHE P06276 1/20 0.34
RIPK1 Q13546 1/20 0.33
ALPL P05186 1/20 0.32
ALPI P09923 1/20 0.32
ALPG P10696 1/20 0.32
TP53 P04637 1/20 0.30
ALOX12 P18054 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15956094 0.81 CES2 (0.49) CES2CES1TP53
SCHEMBL6340967 0.79
SCHEMBL1931609 0.77 CES2 (0.47) CES2CES1BCHERIPK1
SCHEMBL1931608 0.77 CES2 (0.47) CES2CES1BCHERIPK1
SCHEMBL7486005 0.74 STAT3 (0.33)
SCHEMBL5388423 0.73 CES2 (0.67) CES2CES1BCHERIPK1ALPL
SCHEMBL1476095 0.72 MEP1B (0.34) CES2CES1
SCHEMBL2086910 0.72 SLC6A12 (0.33)
SCHEMBL1012189 0.72 CES2 (0.52) CES2CES1
SCHEMBL1012187 0.72 CES2 (0.52) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763539-A1 ANTIBACTERIAL COMPOUNDS Glaxo Group Limited (GB) 2014-08-13 EP disclosed
WO-2013052568-A1 ANTIBACTERIAL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-04-11 WO disclosed