SCHEMBL14846355

SCHEMBL14846355

NC(=S)NNC(=O)COc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.68
MEN1 O00255 9/20 0.65
KMT2A Q03164 9/20 0.65
POLB P06746 4/20 0.65
MAPT P10636 4/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
ADAMTS5 Q9UNA0 2/20 0.58
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
ATM Q13315 1/20 0.56
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
THRB P10828 1/20 0.54
MCL1 Q07820 1/20 0.54
CTDSP1 Q9GZU7 1/20 0.54
ADAMTS4 O75173 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3999404 0.82 ALDH1A1 (0.76) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL2836012 0.82 POLB (0.63) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL31239064 0.80 NPC1 (0.69) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL432126 0.80 CYP19A1 (0.67) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL3740206 0.79 NPC1 (0.63) ALDH1A1MEN1KMT2AL3MBTL1ADAMTS5
SCHEMBL7778609 0.79 ALDH1A1 (0.66) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL3726972 0.79 UBE2N (0.59) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL8626932 0.78 POLB (0.59) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL17988265 0.78 KMT2A (0.68) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL8712014 0.77 ALDH1A1 (0.56) ALDH1A1MEN1KMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2760856-B1 SELECTIVE NR2B ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2016-09-14 EP disclosed
WO-2013049119-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-04 WO disclosed