SCHEMBL148482

SCHEMBL148482

CC(=O)c1ccc(=O)n(-c2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.58
ALDH1A1 P00352 3/20 0.58
HSD17B10 Q99714 2/20 0.58
KDM4E B2RXH2 2/20 0.58
CYP1A2 P05177 1/20 0.58
BLM P54132 1/20 0.58
FGFR1 P11362 1/20 0.48
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GAA P10253 1/20 0.40
KMT2A Q03164 3/20 0.40
TAAR1 Q96RJ0 1/20 0.40
MEN1 O00255 1/20 0.39
HSP90AA1 P07900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL146048 0.85 KDM4E (0.56) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL16474401 0.83 HSD17B10 (0.43) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL16474399 0.83 KMT2A (0.50) ALDH1A1HSD17B10KDM4EMAPTSMN1; SMN2
SCHEMBL10059414 0.82 MAPT (0.61) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL11896477 0.82 KDM4E (0.53) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL11316543 0.82 BLM (0.53) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL13075771 0.81 ALDH1A1 (0.57) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL142307 0.81 KDM4E (0.53) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL16474400 0.81 ALDH1A1 (0.52) HPGDALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL16474398 0.81 KMT2A (0.47) ALDH1A1MAPTLMNAGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 93 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11279733-B2 Peptide antibiotics THE UNIVERSITY OF QUEENSLAND (AU) 2022-03-22 US disclosed
US-20200361994-A1 PEPTIDE ANTIBIOTICS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-11-19 US disclosed
CN-110028442-B Simple preparation method of Perampanel 新发药业有限公司 2020-07-17 CN disclosed
US-10711040-B2 Low substituted polymyxins and compositions thereof XELLIA PHARMACEUTICALS APS (DK) 2020-07-14 US disclosed
US-10640536-B2 Polymyxins, compositions, methods of making and methods of use XELLIA PHARMACEUTICALS APS (DK) 2020-05-05 US disclosed
US-10544161-B2 Anti-fibrotic pyridinones INTERMUNE, INC. (US) 2020-01-28 US disclosed
US-20190321343-A1 Anti-Fibrotic Pyridinones GENENTECH, INC. 2019-10-24 US disclosed
US-10376497-B2 Anti-fibrotic pyridinones INTERMUNE, INC. (US) 2019-08-13 US disclosed
EP-3166960-B1 LOW SUBSTITUTED POLYMYXINS AND COMPOSITIONS THEREOF XELLIA PHARMACEUTICALS APS (DK) 2019-08-07 EP disclosed
US-20190144467-A1 ANTI-FIBROTIC PYRIDINONES GENENTECH, INC. 2019-05-16 US disclosed
US-20090318455-A1 COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY AND FIBROTIC DISORDERS INTERMUNE, INC. (US) 2009-12-24 US disclosed
WO-2009149188-A1 COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY AND FIBROTIC DISORDERS INTERMUNE, INC. (US) 2009-12-10 WO disclosed
EP-1948178-A2 METHODS OF TREATING ATRIAL FIBRILLATION WITH P38 INHIBITOR COMPOUNDS Intermune, Inc. (US) 2008-07-30 EP disclosed
EP-1928454-A2 PYRIDONE DERIVATIVES FOR MODULATING STRESS-ACTIVATED PROTEIN KINASE SYSTEM Intermune, Inc. (US) 2008-06-11 EP disclosed
WO-2007062167-A9 METHOD OF MODULATING STRESS-ACTIVATED PROTEIN KINASE SYSTEM INTERMUNE INC (US) 2007-07-26 WO disclosed
WO-2007062167-A2 METHOD OF MODULATING STRESS-ACTIVATED PROTEIN KINASE SYSTEM INTERMUNE, INC. (US) 2007-05-31 WO disclosed
WO-2007053685-A2 METHODS OF TREATING ATRIAL FIBRILLATION WITH P38 INHIBITOR COMPOUNDS INTERMUNE, INC. (US) 2007-05-10 WO disclosed
WO-2007053685-A2 METHODS OF TREATING ATRIAL FIBRILLATION WITH P38 INHIBITOR COMPOUNDS INTERMUNE, INC. (US) 2007-05-10 WO disclosed
US-20060270612-A1 Method of modulating stress-activated protein kinase system INTERMUNE, INC. 2006-11-30 US disclosed
WO-2006122154-A2 PYRIDONE DERIVATIVES FOR MODULATING STRESS-ACTIVATED PROTEIN KINASE SYSTEM INTERMUNE, INC. (US) 2006-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10544161-B2 Anti-fibrotic pyridinones MMP1, COL1A1, COL2A1 HPGD 298/4885ALDH1A1 529/4885HSD17B10 2171/4885
US-20190321343-A1 Anti-Fibrotic Pyridinones MMP1, COL1A1, COL2A1 HPGD 298/4885ALDH1A1 529/4885HSD17B10 2171/4885
US-10640536-B2 Polymyxins, compositions, methods of making and methods of use C5, HRH3, SGMS1 HPGD 3594/4885ALDH1A1 4877/4885HSD17B10 2236/4885
US-10376497-B2 Anti-fibrotic pyridinones MMP1, COL1A1, COL2A1 HPGD 298/4885ALDH1A1 529/4885HSD17B10 2171/4885
US-20090318455-A1 COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY AND FIBROTIC DISORDERS MAP3K8, MAP3K1, MAP3K6 HPGD 529/4885ALDH1A1 2054/4885HSD17B10 2915/4885
US-20200361994-A1 PEPTIDE ANTIBIOTICS NGLY1, VIP, PEPD HPGD 3755/4885ALDH1A1 4862/4885HSD17B10 4233/4885
US-11279733-B2 Peptide antibiotics NGLY1, VIP, PEPD HPGD 3755/4885ALDH1A1 4862/4885HSD17B10 4233/4885
US-20060270612-A1 Method of modulating stress-activated protein kinase system MAPKAPK2, MAP3K6, MAP4K1 HPGD 995/4885ALDH1A1 3375/4885HSD17B10 3533/4885
US-20190144467-A1 ANTI-FIBROTIC PYRIDINONES MMP1, COL1A1, COL2A1 HPGD 298/4885ALDH1A1 529/4885HSD17B10 2171/4885
US-10711040-B2 Low substituted polymyxins and compositions thereof TLR3, TLR4, TLR5 HPGD 3674/4885ALDH1A1 4882/4885HSD17B10 4006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.