SCHEMBL14852

SCHEMBL14852

Cc1ccc(CNS(C)(=O)=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.61
MEN1 O00255 3/20 0.61
RECQL P46063 2/20 0.56
CA12 O43570 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
ATM Q13315 1/20 0.55
CA9 Q16790 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 4/20 0.53
LMNA P02545 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 1/20 0.51
KDM4E B2RXH2 1/20 0.51
POLB P06746 1/20 0.51
TSHR P16473 1/20 0.51
MAPT P10636 1/20 0.50
CNR2 P34972 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3605081 0.83 KMT2A (0.61) KMT2AMEN1RECQLCA12CA9
SCHEMBL4491485 0.83 KMT2A (0.61) KMT2AMEN1RECQLCA12CA9
SCHEMBL2100494 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9
SCHEMBL6338974 0.81 KMT2A (0.70) KMT2AMEN1RECQLL3MBTL1ALDH1A1
SCHEMBL552189 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9
SCHEMBL7230378 0.81 KMT2A (0.65) KMT2AMEN1RECQLCA12CA9
SCHEMBL5314524 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9
SCHEMBL3599158 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9
SCHEMBL22497546 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9
SCHEMBL14862123 0.81 KMT2A (0.59) KMT2AMEN1RECQLCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 121 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11932613-B2 Process for preparing 1,1,3-trioxo-1,2-benzothiazole-6-carboxamide ADAMA AGAN LTD. (IL) 2024-03-19 US disclosed
US-20230159469-A1 NOVEL PHTHALAZINE DERIVATIVE HAVING ECTONUCLOEOTIDE PYROPHOSPHATASE/PHOSPHODIESTE RASE INHIBITORY ACTIVITY, AND USE THEREOF TXINNO BIOSCIENCE INC. (KR) 2023-05-25 US disclosed
CN-108430981-B Process for preparing 1,1, 3-trioxo-1, 2-benzothiazole-6-carboxamides 阿达玛阿甘股份有限公司 2022-05-10 CN disclosed
CN-108473450-B Process for preparing 1,1, 3-trioxo-1, 2-benzothiazole-6-carboxamides 阿达玛阿甘股份有限公司 2022-05-10 CN disclosed
CN-113089005-B Electrochemical synthesis method of sulfamide 华南理工大学 2022-02-15 CN disclosed
US-20210347746-A1 PROCESS FOR PREPARING 1,1,3-TRIOXO-1,2-BENZOTHIAZOLE-6-CARBOXAMIDE ADAMA AGAN LTD. (IL) 2021-11-11 US disclosed
WO-2021225407-A1 NOVEL PHTHALAZINE DERIVATIVE HAVING ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE INHIBITORY ACTIVITY, AND USE THEREOF 주식회사 티씨노바이오사이언스 (KR) 2021-11-11 WO disclosed
CN-113089005-A Electrochemical synthesis method of sulfamide 华南理工大学 2021-07-09 CN disclosed
EP-3397621-B1 PROCESS FOR PREPARING 1,1,3-TRIOXO-1,2-BENZOTHIAZOLE-6-CARBOXAMIDE ADAMA AGAN LTD (IL) 2020-12-09 EP disclosed
EP-3397620-B1 PROCESS FOR PREPARING 1.1.3-TRIOXO-1.2-BENZOTHIAZOLE-6-CARBOXAMIDE ADAMA AGAN LTD (IL) 2020-11-25 EP disclosed
US-20080113985-A1 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED 2008-05-15 US disclosed
US-20080081809-A1 Novel Compounds KUDOS PHARMACEUTICALS LIMITED (GB) 2008-04-03 US disclosed
US-20080081809-A1 Novel Compounds KUDOS PHARMACEUTICALS LIMITED (GB) 2008-04-03 US disclosed
WO-2008023161-A1 2-METHYLMORPHOLINE PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2008-02-28 WO disclosed
US-20070219228-A1 Aryl substituted imidazonaphthyridines 3M INNOVATIVE PROPERTIES COMPANY 2007-09-20 US disclosed
US-20070219228-A1 Aryl substituted imidazonaphthyridines 3M INNOVATIVE PROPERTIES COMPANY 2007-09-20 US disclosed
US-7271270-B2 High affinity small molecule C5a receptor modulators NEUROGEN CORPORATION (US) 2007-09-18 US disclosed
US-20070213323-A1 NOVEL PYRIDINONE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2-RECEPTORS Janssen Pharmaceuticals, Inc. 2007-09-13 US disclosed
US-20070213323-A1 NOVEL PYRIDINONE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2-RECEPTORS Janssen Pharmaceuticals, Inc. 2007-09-13 US disclosed
WO-2007084413-A2 METHODS FOR TREATING HEPATITIS C PTC THERAPEUTICS, INC. (US) 2007-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210347746-A1 PROCESS FOR PREPARING 1,1,3-TRIOXO-1,2-BENZOTHIAZOLE-6-CARBOXAMIDE TMT1A, TST, CPS1 KMT2A 1010/4885MEN1 3348/4885RECQL 3427/4885
US-20070213323-A1 NOVEL PYRIDINONE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2-RECEPTORS GRM2, GRM1, GRM3 KMT2A 1937/4885MEN1 3509/4885RECQL 962/4885
US-11932613-B2 Process for preparing 1,1,3-trioxo-1,2-benzothiazole-6-carboxamide TMT1A, TST, CPS1 KMT2A 1132/4885MEN1 3249/4885RECQL 3321/4885
US-20080113985-A1 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 KMT2A 4241/4885MEN1 4705/4885RECQL 386/4885
US-20070219228-A1 Aryl substituted imidazonaphthyridines IL2, IRF3, EIF2AK2 KMT2A 3772/4885MEN1 4622/4885RECQL 3346/4885
US-20230159469-A1 NOVEL PHTHALAZINE DERIVATIVE HAVING ECTONUCLOEOTIDE PYROPHOSPHATASE/PHOSPHODIESTE RASE INHIBITORY ACTIVITY, AND USE THEREOF ENPP1, ENPP3, PPA1 KMT2A 3621/4885MEN1 644/4885RECQL 2259/4885
US-20080081809-A1 Novel Compounds SLC10A1, ABCB11, PKD1 KMT2A 3079/4885MEN1 64/4885RECQL 2960/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.