SCHEMBL14865362

SCHEMBL14865362

C[C@@]1(C(=O)NCc2ncc(Nc3c(F)cccc3C(F)(F)F)cc2Cl)CCOC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.37
PTGES O14684 3/20 0.36
PTGS2 P35354 1/20 0.35
CNR2 P34972 4/20 0.34
MAPK8 P45983 2/20 0.34
MAPK9 P45984 2/20 0.34
MAPK10 P53779 2/20 0.34
RAF1 P04049 1/20 0.34
JAK1 P23458 2/20 0.34
JAK3 P52333 2/20 0.34
JAK2 O60674 1/20 0.34
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.34
MAPK14 Q16539 1/20 0.34
NR1I2 O75469 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2809565 0.89 P2RX7 (0.37) P2RX7PTGESPTGS2CNR2MAPK8
SCHEMBL14865294 0.88 P2RX7 (0.36) P2RX7PTGESCNR2MAPK9MAPK10
SCHEMBL2810139 0.85 BDKRB1 (0.36) P2RX7PTGESPTGS2CNR2MAPK8
SCHEMBL185877 0.83 P2RX7 (0.36) P2RX7PTGESPTGS2CNR2MAPK8
SCHEMBL2806537 0.83 P2RX7 (0.34) P2RX7PTGESCNR2MAPK8MAPK9
SCHEMBL2809935 0.82 BDKRB1 (0.38) P2RX7PTGESCNR2RAF1KCNH2
SCHEMBL2807071 0.82 BDKRB1 (0.35) P2RX7PTGESCNR2MAPK8MAPK9
SCHEMBL185684 0.82 BDKRB1 (0.35) P2RX7PTGESCNR2MAPK8MAPK9
SCHEMBL185693 0.81 FGFR4 (0.33) P2RX7PTGESJAK1JAK3JAK2
SCHEMBL14857218 0.81 MAPK7 (0.32) P2RX7PTGESCNR2MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed