SCHEMBL14879545

SCHEMBL14879545

Cc1c(C(F)(F)F)n[nH]c1-c1ccc(NC(=O)c2c(F)cc(F)cc2F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.43
MAPT P10636 1/20 0.43
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HTR1F P30939 1/20 0.39
LRRK2 Q5S007 1/20 0.38
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
IL2 P60568 1/20 0.37
XDH P47989 3/20 0.36
SLC22A12 Q96S37 2/20 0.36
LMNA P02545 3/20 0.36
TSHR P16473 1/20 0.36
EPAS1 Q99814 1/20 0.36
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14879597 0.88 LRRK2 (0.41) POLBMAPTALDH1A1CYP1A2CYP3A4
SCHEMBL14879483 0.84 PTPRC (0.48) MAPTALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL14879594 0.81 RAB9A (0.54) POLBMAPTALDH1A1CYP1A2CYP3A4
SCHEMBL14879421 0.81 P2RX1 (0.40) CSF1RKITKDR
SCHEMBL14879598 0.78 TRPA1 (0.47) CYP1A2IL2LMNAEPAS1HTT
SCHEMBL14879607 0.74 NPC1 (0.45) MAPTALDH1A1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL15578007 0.72 MAPT (0.52) POLBMAPTALDH1A1SMN1; SMN2HSD17B10
SCHEMBL14879553 0.71 GLA (0.38) POLBMAPTKDM4ETSHRKIT
SCHEMBL16008936 0.71 STIM1 (0.52) POLBMAPTALDH1A1CYP1A2CYP3A4
SCHEMBL14879458 0.71 MEN1 (0.46) MAPTALDH1A1SMN1; SMN2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2768810-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2014-08-27 EP disclosed
WO-2013059666-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2013-04-25 WO disclosed