SCHEMBL14891731

SCHEMBL14891731

[CH2]CCCN(C)S(C)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14892638 0.93 MEN1 (0.37) MEN1KMT2A
SCHEMBL14892794 0.91 MEN1 (0.35) MEN1KMT2A
SCHEMBL2248793 0.84
SCHEMBL2853054 0.78 CA2 (0.36)
SCHEMBL11989255 0.77 MEN1 (0.44) MEN1KMT2A
SCHEMBL17327624 0.77 ALDH1A1 (0.43) MEN1KMT2A
SCHEMBL4374311 0.77 MEN1 (0.44) MEN1KMT2A
SCHEMBL23838730 0.75 MEN1 (0.38) MEN1KMT2A
SCHEMBL12967466 0.75 DNM1 (0.46) MEN1KMT2A
SCHEMBL4374314 0.75 MEN1 (0.43) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9187450-B2 Substituted pyridine compound DAIICHI SANKYO COMPANY, LIMITED (JP) 2015-11-17 US disclosed
EP-2592076-B1 SUBSTITUTED PYRIDINE COMPOUND DAIICHI SANKYO CO LTD (JP) 2015-05-13 EP disclosed
CN-103221405-B Substituted pyridine compound DAIICHI SANKYO CO LTD 2015-04-22 CN disclosed
US-20140213549-A9 Substituted Pyridine Compound UBE INDUSTRIES, LTD. (JP) 2014-07-31 US disclosed
US-20140005143-A2 Substituted PyridineCompound DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-01-02 US disclosed
CN-103221405-A Substituted pyridine compound DAIICHI SANKYO CO LTD 2013-07-24 CN disclosed
EP-2592076-A1 SUBSTITUTED PYRIDINE COMPOUND DAIICHI SANKYO COMPANY, LIMITED (JP) 2013-05-15 EP disclosed
US-20130109653-A1 Substituted Pyridine Compound UBE INDUSTRIES, LTD. (JP) 2013-05-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140213549-A9 Substituted Pyridine Compound CETP, MTTP, PRCP MEN1 3088/4885KMT2A 1200/4885
US-20140005143-A2 Substituted PyridineCompound CETP, MTTP, CES1 MEN1 3487/4885KMT2A 1462/4885
US-20130109653-A1 Substituted Pyridine Compound CETP, MTTP, PRCP MEN1 3088/4885KMT2A 1200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.