SCHEMBL14899552

SCHEMBL14899552

CCOC(=O)C1=NCCc2cc(OC)c(C)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.49
HSD17B10 Q99714 2/20 0.49
KMT2A Q03164 2/20 0.49
MAOA P21397 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.46
KCNK3 O14649 1/20 0.46
NPSR1 Q6W5P4 1/20 0.44
RAD52 P43351 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
GLA P06280 1/20 0.38
RCE1 Q9Y256 1/20 0.38
HSD17B2 P37059 1/20 0.38
LMNA P02545 1/20 0.38
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1202228 0.92 KDM4E (0.57) KDM4EHSD17B10KMT2AMAOAALDH1A1
SCHEMBL1143224 0.83 KDM4E (0.44) KDM4EHSD17B10KMT2AMAOAALDH1A1
SCHEMBL10515648 0.80 KDM4E (0.44) KDM4EALDH1A1MAPTGAAHPGD
SCHEMBL1143122 0.80 KDM4E (0.46) KDM4EHSD17B10KMT2AALDH1A1MAPT
SCHEMBL4123425 0.75 TSHR (0.43) KDM4EKMT2AALDH1A1MAPTGAA
SCHEMBL10517138 0.74 MAPT (0.43) KDM4EKMT2AMAPTNPSR1CYP1A2
SCHEMBL12071541 0.74 MAOA (0.81) KDM4EHSD17B10MAOAALDH1A1MAPT
SCHEMBL4117558 0.74 ALDH1A1 (0.51) KDM4EHSD17B10KMT2AALDH1A1MAPT
SCHEMBL18070225 0.72 UGCG (0.47) KDM4EHSD17B10KMT2AALDH1A1MAPT
SCHEMBL27669711 0.70 KDM4E (0.48) KDM4EHSD17B10KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8431564-B2 Ring-annulated dihydropyrrolo[2,1-α]isoquinolines MERCK SHARP & DOHME B.V. (NL) 2013-04-30 US disclosed