SCHEMBL14919381

SCHEMBL14919381

CCOC(OCC)C1C(=O)c2cc(OC)ccc2OC12CCN(C(=O)O)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.40
KLK7 P49862 1/20 0.40
ALDH1A1 P00352 11/20 0.39
HPGD P15428 8/20 0.39
GAA P10253 7/20 0.39
CASP1 P29466 4/20 0.39
HSD17B10 Q99714 4/20 0.39
HTR2C P28335 1/20 0.37
PPIB P23284 1/20 0.37
GLA P06280 5/20 0.37
CASP7 P55210 2/20 0.37
KMT2A Q03164 1/20 0.37
CYP19A1 P11511 2/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
THRB P10828 1/20 0.35
POLB P06746 1/20 0.35
ABCB1 P08183 1/20 0.35
AR P10275 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2595165 0.89 KMT2A (0.40) KDM4EKLK7ALDH1A1HPGDGAA
SCHEMBL2592656 0.88 HSD11B1 (0.39) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL2590155 0.85 KMT2A (0.35) KDM4EALDH1A1KMT2A
SCHEMBL14919186 0.82 HDAC8 (0.34) KDM4EALDH1A1GAAHSD17B10KMT2A
SCHEMBL2594530 0.77 KMT2A (0.39) ALDH1A1GAAKMT2ASMN1; SMN2POLB
SCHEMBL2588272 0.77 GPR119 (0.40) KMT2A
SCHEMBL2592446 0.74 GPR119 (0.38) KDM4EKMT2A
SCHEMBL2594720 0.72 ALDH1A1 (0.59) KDM4EKLK7ALDH1A1HPGDGAA
SCHEMBL2586856 0.72 GPR119 (0.40) KMT2A
SCHEMBL14972718 0.69 EPHX2 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013067248-A1 BENZOXAZINES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-05-10 WO disclosed