SCHEMBL14920974

SCHEMBL14920974

COC(=O)c1ccc(NCc2ccc(OC)cc2)nc1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 7/20 0.64
HDAC1 Q13547 4/20 0.64
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
KMT2A Q03164 1/20 0.60
MAPT P10636 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
HDAC3 O15379 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
GABRA5 P31644 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11563704 0.89 VNN1 (0.64) VNN1HDAC1NPC1RAB9AKMT2A
SCHEMBL30465779 0.88 VNN1 (0.70) VNN1HDAC1NPC1RAB9AKMT2A
SCHEMBL11567319 0.88 ALDH1A1 (0.61) VNN1HDAC1CA1CA2GABRA5
SCHEMBL22084214 0.86 VNN1 (0.57) VNN1HDAC1NPC1RAB9AMAPT
SCHEMBL20722658 0.86 CA1 (0.62) VNN1HDAC1CA1CA2HDAC3
SCHEMBL17602245 0.84 HDAC1 (0.57) VNN1HDAC1NPC1RAB9AKMT2A
SCHEMBL2308761 0.82 NPC1 (0.68) VNN1HDAC1NPC1RAB9AKMT2A
SCHEMBL10255569 0.81 HDAC1 (0.67) VNN1HDAC1NPC1RAB9AKMT2A
SCHEMBL16211422 0.81 RAB9A (0.54) VNN1NPC1RAB9AKMT2AMAPT
SCHEMBL18424186 0.81 SMN1; SMN2 (0.56) HDAC1NPC1RAB9ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9145354-B2 Pharmaceutical compounds ASTEX THERAPEUTICS LIMITED (GB) 2015-09-29 US disclosed
US-20150051199-A1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2015-02-19 US disclosed
EP-2773615-A1 PHARMACEUTICAL COMPOUNDS Astex Therapeutics Limited (GB) 2014-09-10 EP disclosed
WO-2013064543-A1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2013-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150051199-A1 PHARMACEUTICAL COMPOUNDS NR1H4, HAVCR2, NR1H3 VNN1 3177/4885HDAC1 1052/4885NPC1 66/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.