SCHEMBL14922282

SCHEMBL14922282

CN1CCN(c2ccc(F)c(F)c2F)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
POLB P06746 1/20 0.47
ADRA2C P18825 1/20 0.44
KDM4E B2RXH2 4/20 0.43
MAPT P10636 4/20 0.43
RAD52 P43351 1/20 0.43
PHGDH O43175 1/20 0.43
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
DRD1 P21728 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2A P28223 1/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13382891 0.82 DRD2 (0.53) ALDH1A1L3MBTL1POLBADRA2CKDM4E
SCHEMBL16514423 0.81 ALDH1A1 (0.62) ALDH1A1L3MBTL1POLBADRA2CKDM4E
SCHEMBL28296311 0.79 PHGDH (0.40) ALDH1A1L3MBTL1POLBMAPTPHGDH
SCHEMBL4794953 0.77 PDE7A (0.38) ALDH1A1POLBKDM4EMAPTPHGDH
SCHEMBL9657066 0.77 RAD52 (0.44) ALDH1A1POLBKDM4EMAPTRAD52
SCHEMBL8191985 0.76 HTR1A (0.46) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2894409 0.76 ALDH1A1 (0.60) ALDH1A1L3MBTL1POLBADRA2CKDM4E
SCHEMBL8275465 0.76 POLB (0.65) ALDH1A1L3MBTL1POLBKDM4EMAPT
SCHEMBL6924885 0.74 ALDH1A1 (0.69) ALDH1A1L3MBTL1POLBKDM4EMAPT
SCHEMBL19262490 0.74 ALDH1A1 (0.64) ALDH1A1L3MBTL1POLBADRA2CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed