SCHEMBL14922305

SCHEMBL14922305

COCCOc1ccc(N(C)CCN(C)C)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.45
THRB P10828 1/20 0.45
PDK2 Q15119 2/20 0.38
BRAF P15056 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
HRH3 Q9Y5N1 3/20 0.35
TNF P01375 1/20 0.34
IL6 P05231 1/20 0.34
CACNA1B Q00975 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
LTA4H P09960 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14922255 0.86 THRA (0.38) THRATHRBPDK2KDM4EALDH1A1
SCHEMBL8257891 0.75 MAOA (0.39) THRATHRBKDM4EALDH1A1
SCHEMBL10352711 0.74 FFAR4 (0.43) THRATHRBALDH1A1
SCHEMBL10104423 0.73 CRHR1 (0.37) BRAFSMN1; SMN2
SCHEMBL12875595 0.73 EPHX2 (0.46) THRATHRB
SCHEMBL1407867 0.72 GAA (0.47) BRAFKDM4EALDH1A1HRH3
SCHEMBL13812978 0.71 GLA (0.43) BRAF
SCHEMBL6718732 0.71 THRA (0.48) THRATHRBPDK2KDM4EALDH1A1
SCHEMBL25919977 0.71 THRA (0.40) THRATHRBPDK2KDM4EALDH1A1
SCHEMBL14430363 0.70 THRA (0.50) THRATHRBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed