SCHEMBL14922307

SCHEMBL14922307

CN1CCN(c2ccc(CO)cc2C(F)(F)F)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.49
CHKA P35790 1/20 0.47
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
CDK4 P11802 3/20 0.42
CCND3 P30281 3/20 0.42
GSK3B P49841 3/20 0.42
PIM1 P11309 2/20 0.42
CCNA2 P20248 7/20 0.42
CDK2 P24941 7/20 0.42
CCNA1 P78396 7/20 0.42
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SRPK1 Q96SB4 1/20 0.40
MTOR P42345 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12141731 0.87 ASIC3 (0.50) ASIC3PDE3BPDE3ACDK4CCND3
SCHEMBL251465 0.85 ASIC3 (0.49) ASIC3CHKAPDE3BPDE3ACDK4
SCHEMBL10088914 0.85 NOTUM (0.47)
SCHEMBL12141713 0.80 AKR1C3 (0.48) ASIC3PDE3BPDE3ACCNA2CDK2
SCHEMBL250792 0.80 TRPV1 (0.46) ASIC3PDE3BPDE3ACDK4CCND3
SCHEMBL24309870 0.80 ASIC3 (0.52) ASIC3PDE3BPDE3ACDK4CCND3
SCHEMBL14922289 0.80 CHKA (0.50) CHKAALDH1A1L3MBTL1
SCHEMBL14922283 0.78 CHKA (0.51) CHKAALDH1A1L3MBTL1
SCHEMBL12017807 0.78 ADRB2 (0.55) ASIC3PDE3BPDE3ACDK4CCND3
SCHEMBL29959068 0.77 MAPT (0.59) ASIC3PDE3BPDE3ACDK4CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed