SCHEMBL14922283

SCHEMBL14922283

Cc1cc(CO)ccc1N1CCN(C)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.51
MAPT P10636 5/20 0.42
GAA P10253 3/20 0.42
RAD52 P43351 2/20 0.42
GFER P55789 1/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 3/20 0.41
POLB P06746 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KMT2A Q03164 2/20 0.40
PTK2B Q14289 2/20 0.40
MEN1 O00255 1/20 0.40
THRB P10828 1/20 0.40
NR4A1 P22736 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
JAK3 P52333 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14554255 0.85 HTR1A (0.47) MAPTGAARAD52GFERALDH1A1
SCHEMBL10088504 0.85 ALDH1A1 (0.53) CHKAMAPTGAARAD52GFER
SCHEMBL6111730 0.84 RAD52 (0.61) MAPTGAARAD52GFERALDH1A1
SCHEMBL29493256 0.83 MAPT (0.45) CHKAMAPTGAARAD52GFER
SCHEMBL14922289 0.82 CHKA (0.50) CHKAMAPTRAD52ALDH1A1KDM4E
SCHEMBL14687616 0.82 HTR3A (0.56) HTR1AHTR3A
SCHEMBL14922273 0.80 DRD2 (0.55) CHKAMAPTALDH1A1KDM4EPOLB
SCHEMBL14922307 0.78 ASIC3 (0.49) CHKAALDH1A1L3MBTL1
SCHEMBL29287728 0.77 CYP2D6 (0.39) MAPTGAARAD52GFERALDH1A1
SCHEMBL7923952 0.77 HTR1A (0.58) MAPTGAAALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed