SCHEMBL14923013

SCHEMBL14923013

C[C@H]1CC(c2ccc(OC(F)F)c(F)c2)=NN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.41
HRH3 Q9Y5N1 1/20 0.36
MAOA P21397 2/20 0.34
MAOB P27338 1/20 0.34
KCNH2 Q12809 3/20 0.34
GRIN2B Q13224 3/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
PDE2A O00408 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14922983 0.79 DRD1 (0.38) LMNA
SCHEMBL14596843 0.67 ESR2 (0.41) GRM2KCNH2GRIN2BPDE2A
SCHEMBL28052513 0.66 SMN1; SMN2 (0.46) GRM2KCNH2GRIN2BPDE4APDE4B
SCHEMBL10072935 0.65 RAB9A (0.51) MAOAMAOBLMNACYP1A2HPGD
SCHEMBL7916857 0.64 KIF11 (0.47) GRIN2B
SCHEMBL9220447 0.64 CYP17A1 (0.46) GRM2KCNH2GRIN2BLMNA
SCHEMBL20529059 0.64 MAOA (0.44) GRM2MAOAMAOBPDE4APDE4B
SCHEMBL30244557 0.64 GRIN2B (0.40) GRM2KCNH2GRIN2BPDE4APDE4B
SCHEMBL18134246 0.63 FASN (0.39) GRM2PDE4BPDE4DCYP2C9CYP2C19
SCHEMBL9226568 0.63 PDE3B (0.39) GRM2GRIN2BPDE3BPDE3ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118067-B1 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS SIENA BIOTECH SPA (IT) 2013-05-08 EP disclosed