SCHEMBL14928512

SCHEMBL14928512

CC(C)[C@@H](C1CC1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
LMNA P02545 3/20 0.44
ALDH1A1 P00352 5/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
KMT2A Q03164 2/20 0.41
GAA P10253 1/20 0.41
CASP3 P42574 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16169047 1.00 TDP1 (0.45) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL14928513 0.93 ALDH1A1 (0.44) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL16169045 0.86 TDP1 (0.42) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL15081302 0.86 TDP1 (0.42) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL16169030 0.83 TDP1 (0.44) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL16164903 0.79 LMNA (0.46) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL16164902 0.79 LMNA (0.46) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL16169049 0.78 TSHR (0.42) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL6925075 0.74 ALDH1A1 (0.49) TDP1LMNAALDH1A1HTTNPC1
SCHEMBL6925072 0.74 ALDH1A1 (0.49) TDP1LMNAALDH1A1HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051310-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2015-06-09 US disclosed
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2014-10-16 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK TDP1 2598/4885LMNA 3649/4885ALDH1A1 1638/4885
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, BTK, NOX4 TDP1 1179/4885LMNA 4440/4885ALDH1A1 982/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.