SCHEMBL14931121

SCHEMBL14931121

CC(C)(C)OC(=O)N[C@H](CN1C(=O)c2ccccc2C1=O)c1ccsc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.41
CTSK P43235 2/20 0.41
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP3 P08254 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
MALT1 Q9UDY8 1/20 0.38
SCN9A Q15858 3/20 0.38
KMT2A Q03164 3/20 0.37
PTPRB P23467 1/20 0.37
AKT1 P31749 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.36
CCKAR P32238 1/20 0.35
CCKBR P32239 1/20 0.35
MEN1 O00255 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14908706 0.87 CTSK (0.47) CTSSCTSKMALT1SCN9AKMT2A
SCHEMBL3374003 0.87 CTSK (0.47) CTSSCTSKMALT1SCN9AKMT2A
SCHEMBL3760185 0.87 CTSK (0.47) CTSSCTSKMALT1SCN9AKMT2A
SCHEMBL14911465 0.83 ALDH1A1 (0.42) KMT2AALDH1A1MEN1THRB
SCHEMBL34471389 0.83 ALDH1A1 (0.46) CTSSCTSKMMP1MMP2MMP3
SCHEMBL30109123 0.82 CTSS (0.41) CTSSCTSKKMT2AAKT1ALDH1A1
SCHEMBL5576694 0.81 KMT2A (0.43) CTSSCTSKKMT2AALDH1A1MEN1
SCHEMBL30109325 0.81 POLB (0.48) KMT2AALDH1A1ATMMEN1
SCHEMBL30109136 0.81 POLB (0.48) KMT2AALDH1A1ATMMEN1
SCHEMBL23017648 0.81 KMT2A (0.43) KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed
CN-102958918-A Novel nicotinamide derivatives or salts thereof FUJIFILM CORP 2013-03-06 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK CTSS 3435/4885CTSK 3872/4885MMP1 2912/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.