SCHEMBL14939349

SCHEMBL14939349

COc1ccccc1CN1CCN(C2(c3cccc(C)c3)Cc3ccccc3C2=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
CXCR4 P61073 1/20 0.43
DRD2 P14416 4/20 0.43
DRD4 P21917 3/20 0.43
HRH2 P25021 1/20 0.41
DRD3 P35462 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CHRM3 P20309 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 3/20 0.40
CYP2D6 P10635 2/20 0.40
TSHR P16473 2/20 0.40
HTR1A P08908 1/20 0.40
HTR2B P41595 1/20 0.40
HTR7 P34969 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939017 0.90 HTR7 (0.48) ALDH1A1MAPTHTTDRD2DRD4
SCHEMBL14939959 0.90 MEN1 (0.48) ALDH1A1DRD2DRD4HRH2DRD3
SCHEMBL14939342 0.90 CYP2D6 (0.48) ALDH1A1DRD2DRD4HRH2DRD3
SCHEMBL14939091 0.88 KMT2A (0.42) ALDH1A1MAPTHTTDRD2DRD4
SCHEMBL14939559 0.88 KMT2A (0.42) ALDH1A1MAPTHTTDRD2DRD4
SCHEMBL14939089 0.88 KMT2A (0.42) ALDH1A1MAPTHTTDRD2DRD4
SCHEMBL14939609 0.84 NPSR1 (0.52) ALDH1A1MAPTHTTCXCR4DRD2
SCHEMBL14939466 0.84 NPSR1 (0.54) ALDH1A1MAPTHTTDRD2CHRM3
SCHEMBL14939480 0.84 NPSR1 (0.48) ALDH1A1MAPTHTTDRD2CHRM3
SCHEMBL14939908 0.84 SIGMAR1 (0.51) ALDH1A1MAPTDRD2CHRM3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed