SCHEMBL14939017

SCHEMBL14939017

COc1cccc(C2(N3CCN(Cc4ccccc4OC)CC3)Cc3ccccc3C2=O)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.48
DRD4 P21917 2/20 0.46
HTT P42858 2/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 1/20 0.42
DRD2 P14416 2/20 0.41
HRH2 P25021 1/20 0.41
DRD3 P35462 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CHRM3 P20309 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
SIGMAR1 Q99720 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939349 0.90 ALDH1A1 (0.46) HTR7DRD4HTTALDH1A1KDM4E
SCHEMBL14938846 0.90 ALDH1A1 (0.41) HTR7HTTALDH1A1KDM4EMEN1
SCHEMBL14939959 0.90 MEN1 (0.48) HTR7DRD4ALDH1A1KDM4ETSHR
SCHEMBL14939342 0.90 CYP2D6 (0.48) HTR7DRD4ALDH1A1TSHRMEN1
SCHEMBL14939907 0.87 SIGMAR1 (0.55) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL14940301 0.87 SIGMAR1 (0.55) HTTALDH1A1DRD2CHRM3HTR2A
SCHEMBL14939591 0.85 SIGMAR1 (0.50) ALDH1A1KDM4EMEN1KMT2ADRD2
SCHEMBL14939450 0.84 NPSR1 (0.52) HTR7DRD4HTTALDH1A1KDM4E
SCHEMBL14939836 0.83 TACR1 (0.45) DRD4ALDH1A1KDM4EMEN1KMT2A
SCHEMBL14939908 0.82 SIGMAR1 (0.51) ALDH1A1KDM4EMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed