SCHEMBL14939375

SCHEMBL14939375

O=C1c2ccccc2C(=O)C1(Br)c1cccc(N2CCOCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
KMO O15229 1/20 0.46
PSMD14 O00487 1/20 0.45
PDK2 Q15119 1/20 0.44
AGXT P21549 1/20 0.44
MAPT P10636 3/20 0.44
PDGFRB P09619 1/20 0.43
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
BRD4 O60885 1/20 0.42
CREBBP Q92793 1/20 0.42
PIK3C3 Q8NEB9 2/20 0.41
KIF11 P52732 1/20 0.41
TDP2 O95551 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939345 0.87 MAPT (0.46) PDK2AGXTMAPTALDH1A1MEN1
SCHEMBL14939995 0.86 MAPT (0.45) PDK2AGXTMAPTALDH1A1MEN1
SCHEMBL14939704 0.84 ADRA2C (0.48) LMNAPDK2AGXTMAPTKMT2A
SCHEMBL14938965 0.74 NPSR1 (0.67) LMNAAGXTMAPTALDH1A1KIF11
SCHEMBL27329825 0.72 LMNA (0.71) LMNAKMOAGXTMAPTALDH1A1
SCHEMBL4699438 0.71 AGXT (0.54) LMNAKMOAGXTMAPTALDH1A1
SCHEMBL14940158 0.70 NPSR1 (0.53) LMNAMAPTALDH1A1SMN1; SMN2MEN1
SCHEMBL14939632 0.70 CA1 (0.43) MAPTALDH1A1SMN1; SMN2RAB9ATDP1
SCHEMBL14939727 0.69 CYP3A4 (0.52) LMNAKMOPSMD14AGXTMAPT
SCHEMBL14973406 0.69 PSMD14 (0.68) LMNAPSMD14PDK2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed