SCHEMBL14939451

SCHEMBL14939451

O=C1c2ccccc2C(=O)C1(Br)c1cccc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.42
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 3/20 0.42
HTT P42858 2/20 0.42
THRB P10828 1/20 0.42
CYP2D6 P10635 1/20 0.41
BACE1 P56817 2/20 0.41
ALOX12 P18054 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CA7 P43166 1/20 0.41
RECQL P46063 1/20 0.41
CA9 Q16790 1/20 0.41
EHMT2 Q96KQ7 1/20 0.41
S100A4 P26447 2/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940158 0.80 NPSR1 (0.53) MAPTALDH1A1NPSR1CYP2D6BACE1
SCHEMBL14939632 0.80 CA1 (0.43) MAPTALDH1A1CYP2D6BACE1ALOX12
SCHEMBL14938923 0.80 MAPT (0.43) MAPTALDH1A1NPSR1HTTTHRB
SCHEMBL14940123 0.79 ALDH1A1 (0.47) MAPTALDH1A1NPSR1HTTTHRB
SCHEMBL14939057 0.78 ALDH1A1 (0.52) MAPTALDH1A1HTTTHRBCYP2D6
SCHEMBL14939165 0.75 MAPT (0.49) MAPTMAOBKDM4EAPAF1TDP2
SCHEMBL14939787 0.75 CYP2D6 (0.38) MAPTALDH1A1NPSR1THRBCYP2D6
SCHEMBL14939005 0.75 KMT2A (0.49) MAPTALDH1A1CYP2D6BACE1CA1
SCHEMBL14939783 0.74 CASP6 (0.40) MAPTALDH1A1NPSR1HTTTHRB
SCHEMBL14939711 0.73 CYP2D6 (0.42) ALDH1A1CYP2D6BACE1ALOX12L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed