SCHEMBL14939711

SCHEMBL14939711

O=C1c2ccccc2C(=O)C1(Br)c1ccc2ccccc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
TSHR P16473 1/20 0.42
ALOX12 P18054 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
CA7 P43166 1/20 0.42
RECQL P46063 1/20 0.42
BACE1 P56817 1/20 0.42
CA9 Q16790 1/20 0.42
EHMT2 Q96KQ7 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GSTP1 P09211 1/20 0.41
HDAC4 P56524 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
SLC6A4 P31645 5/20 0.38
SLC6A3 Q01959 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939057 0.76 ALDH1A1 (0.52) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939461 0.75 CA1 (0.46) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939632 0.74 CA1 (0.43) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14940158 0.74 NPSR1 (0.53) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939402 0.73 CYP2D6 (0.49) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14940123 0.73 ALDH1A1 (0.47) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939593 0.73 CYP2D6 (0.45) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939451 0.73 MAPT (0.42) CYP2D6ALDH1A1CA1CA2TSHR
SCHEMBL14939005 0.73 KMT2A (0.49) CYP2D6ALDH1A1CA1CA2MAPK1
SCHEMBL14939588 0.69 ALDH1A1 (0.50) CYP2D6ALDH1A1CA1CA2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed