SCHEMBL14939005

SCHEMBL14939005

COc1cccc(C2(Br)C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
GAA P10253 1/20 0.49
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA4 P22748 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
MAPT P10636 4/20 0.43
ACHE P22303 1/20 0.43
KDM1A O60341 1/20 0.43
BACE1 P56817 1/20 0.43
BACE2 Q9Y5Z0 1/20 0.43
MAOB P27338 1/20 0.43
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939566 0.82 CA1 (0.56) KMT2AMEN1GAACA1CA2
SCHEMBL14939682 0.81 KMT2A (0.46) KMT2AMEN1GAACA1CA2
SCHEMBL14939090 0.80 CA1 (0.43) KMT2AMEN1GAACA1CA2
SCHEMBL14940158 0.80 NPSR1 (0.53) KMT2AMEN1GAACA1CA2
SCHEMBL14940276 0.77 PPIB (0.43) KMT2AMEN1GAAMAPTKDM1A
SCHEMBL14939632 0.76 CA1 (0.43) GAACA1CA2CA4CA7
SCHEMBL14939451 0.75 MAPT (0.42) GAACA1CA2CA7CA9
SCHEMBL14939057 0.74 ALDH1A1 (0.52) KMT2AMEN1GAACA1CA2
SCHEMBL14939711 0.73 CYP2D6 (0.42) CA1CA2CA7CA9BACE1
SCHEMBL7315657 0.72 PDK2 (0.51) KMT2AMEN1GAAACHEKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed