SCHEMBL14939485

SCHEMBL14939485

COc1ccc2c(c1)CC(c1ccccc1)(N1CCN(Cc3ccccc3)CC1)C2=O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.51
DRD2 P14416 2/20 0.51
HTR2A P28223 2/20 0.51
HTR2C P28335 2/20 0.51
HTR2B P41595 2/20 0.51
ACHE P22303 4/20 0.50
BACE1 P56817 1/20 0.50
NPSR1 Q6W5P4 2/20 0.49
LMNA P02545 1/20 0.47
HTR1A P08908 2/20 0.45
HTR7 P34969 2/20 0.45
HTR6 P50406 2/20 0.45
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
PAX8 Q06710 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940496 0.93 ACHE (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14938869 0.89 SIGMAR1 (0.48) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14940301 0.89 SIGMAR1 (0.55) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939400 0.86 NPSR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939907 0.84 SIGMAR1 (0.55) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939175 0.84 NPSR1 (0.64) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939625 0.84 NPSR1 (0.64) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14940373 0.84 NPSR1 (0.64) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14940098 0.84 NPSR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939880 0.84 NPSR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed