SCHEMBL14940301

SCHEMBL14940301

COc1cccc(C2(N3CCN(Cc4ccccc4)CC3)Cc3ccccc3C2=O)c1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.55
NPSR1 Q6W5P4 1/20 0.51
DRD2 P14416 3/20 0.50
HTR2A P28223 3/20 0.50
HTR2C P28335 3/20 0.50
HTR2B P41595 3/20 0.50
ALDH1A1 P00352 2/20 0.47
ALDH3A1 P30838 1/20 0.47
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
ACHE P22303 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939907 0.96 SIGMAR1 (0.55) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14939591 0.93 SIGMAR1 (0.50) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14939908 0.90 SIGMAR1 (0.51) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14940465 0.89 SIGMAR1 (0.50) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939485 0.89 SIGMAR1 (0.51) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14940496 0.88 ACHE (0.52) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14939017 0.87 HTR7 (0.48) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14938846 0.87 ALDH1A1 (0.41) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939777 0.86 NPSR1 (0.54) SIGMAR1NPSR1DRD2HTR2AHTR2C
SCHEMBL14939466 0.86 NPSR1 (0.54) SIGMAR1NPSR1DRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed