SCHEMBL14938869

SCHEMBL14938869

COc1ccc(CN2CCN(C3(c4ccccc4)Cc4cc(F)ccc4C3=O)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.48
DRD2 P14416 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TACR1 P25103 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940346 0.94 SIGMAR1 (0.44) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939880 0.90 NPSR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939744 0.89 LMNA (0.45) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939485 0.89 SIGMAR1 (0.51) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939836 0.86 TACR1 (0.45) DRD2CHRM3TACR1
SCHEMBL14940059 0.85 NPSR1 (0.49) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14940496 0.84 ACHE (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939526 0.84 NPSR1 (0.46) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939854 0.84 CHRM2 (0.43) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14939469 0.83 SIGMAR1 (0.50) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed