SCHEMBL14944722

SCHEMBL14944722

COc1ccnc(Cn2c3c([nH]c2=O)C(N)NC(n2cccn2)=N3)c1OC

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
USP1 O94782 5/20 0.34
HCRTR1 O43613 11/20 0.33
HCRTR2 O43614 10/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
ADORA1 P30542 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20343814 0.80 USP1 (0.37) USP1ADORA1TLR7
SCHEMBL14944713 0.75 ADORA1 (0.35) USP1HCRTR1HCRTR2ADORA1TLR7
SCHEMBL14944715 0.73 TLR7 (0.41) USP1HCRTR1HCRTR2ADORA1TLR7
SCHEMBL16206183 0.72 TLR7 (0.42) USP1ADORA1TLR7
SCHEMBL14944647 0.59 TLR7 (0.41) TLR7
SCHEMBL20343751 0.58 PNP (0.38) TLR7
SCHEMBL20343763 0.57 TLR7 (0.42) ADORA1TLR7
SCHEMBL20134287 0.57 GRIN1 (0.57) GRIN1GRIN2B
SCHEMBL2690888 0.57 RAB9A (0.41) HSP90AA1HSP90AB1TLR7
SCHEMBL17434630 0.57 RAB9A (0.41) HSP90AA1HSP90AB1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776439-B1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN SCIENCES IRELAND UC (IE) 2018-07-04 EP disclosed
WO-2013068438-A1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN R&D IRELAND (IE) 2013-05-16 WO disclosed