SCHEMBL14947855

SCHEMBL14947855

CCCC[C@H](NC(=O)[C@@H](NC(=O)[C@]1(C)CCC/C=C\CCCC(C)(C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)C(=O)[C@H](CCC(N)=O)NN1)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.47
ESR1 P03372 2/20 0.47
EIF4E P06730 4/20 0.47
EIF4EBP1 Q13541 4/20 0.47
KRAS P01116 4/20 0.47
MDM4 O15151 4/20 0.46
MDM2 Q00987 4/20 0.46
ESR2 Q92731 1/20 0.45
PCSK9 Q8NBP7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16975610 0.96 MDM4 (0.43) MCL1ESR1EIF4EEIF4EBP1KRAS
SCHEMBL14947860 0.94 MDM4 (0.43) MCL1ESR1EIF4EEIF4EBP1KRAS
SCHEMBL14947863 0.89 ESR1 (0.40) MCL1ESR1EIF4EEIF4EBP1KRAS
SCHEMBL14948248 0.89 ESR1 (0.40) MCL1ESR1EIF4EEIF4EBP1KRAS
SCHEMBL15183813 0.70 MDM2 (0.66) ESR1EIF4EEIF4EBP1MDM4MDM2
SCHEMBL16975828 0.69 ESR1 (0.34) MCL1ESR1EIF4EEIF4EBP1MDM4
SCHEMBL14950915 0.69 EIF4E (0.38) MCL1ESR1EIF4EEIF4EBP1MDM4
SCHEMBL19760420 0.69 ESR1 (0.52) ESR1KRASMDM4MDM2ESR2
SCHEMBL17568833 0.65 ESR1 (0.62) MCL1ESR1EIF4EEIF4EBP1KRAS
SCHEMBL17880428 0.65 MAFG (0.53) ESR1KRASESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096684-B2 Peptidomimetic macrocycles AILERON THERAPEUTICS, INC. (US) 2015-08-04 US disclosed
US-20130123169-A1 PEPTIDOMIMETIC MACROCYCLES AILERON THERAPEUTICS, INC. (US) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123169-A1 PEPTIDOMIMETIC MACROCYCLES GHRHR, GHSR, GHITM MCL1 677/4885ESR1 470/4885EIF4E 1654/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.