SCHEMBL14958727

SCHEMBL14958727

Cc1cc(O)cc(C)c1S(=O)(=O)N(C)CCC(=O)Nc1ccc(N2CCCC(N3CCCCC3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.45
TP53 P04637 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 8/20 0.44
KDM4E B2RXH2 7/20 0.44
BDKRB1 P46663 4/20 0.43
HTT P42858 1/20 0.42
KMT2A Q03164 6/20 0.42
MAPT P10636 6/20 0.42
GAA P10253 5/20 0.42
MEN1 O00255 4/20 0.42
MAPK1 P28482 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
USP2 O75604 3/20 0.42
RAD52 P43351 2/20 0.42
GFER P55789 2/20 0.42
ALOX15 P16050 1/20 0.42
NR4A1 P22736 1/20 0.42
MCL1 Q07820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3440208 0.89 BDKRB1 (0.54) ALDH1A1KDM4EBDKRB1KMT2AMAPT
SCHEMBL15372649 0.83 BDKRB1 (0.47) SMN1; SMN2TP53NPC1RAB9AALDH1A1
SCHEMBL3440537 0.82 BDKRB1 (0.59) NPC1RAB9ABDKRB1GAAMAPK1
SCHEMBL14958754 0.82 MAPT (0.54) SMN1; SMN2TP53NPC1RAB9AALDH1A1
SCHEMBL10118727 0.80 BDKRB1 (0.59) BDKRB1KMT2AMAPTMEN1GFER
SCHEMBL3439589 0.79 BDKRB1 (0.49) ALDH1A1KDM4EBDKRB1KMT2AMAPT
SCHEMBL14958780 0.79 BDKRB1 (0.60) BDKRB1KMT2AGFERHRH3
SCHEMBL3440434 0.79 BDKRB1 (0.54) BDKRB1KMT2AMEN1
SCHEMBL3440299 0.78 L3MBTL1 (0.39) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL12914508 0.78 POLB (0.55) SMN1; SMN2NPC1RAB9ABDKRB1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402329-B1 Analgetic phenylsulphonamides BOEHRINGER INGELHEIM INT (DE) 2013-05-22 EP disclosed