SCHEMBL1495894

SCHEMBL1495894

CC(O)C(C)Oc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
GAA P10253 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 1/20 0.40
CA4 P22748 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.40
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
CYP2D6 P10635 1/20 0.39
ADRB3 P13945 1/20 0.39
CHRNB4 P30926 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385111 0.92 LTA4H (0.48) LMNAGAACYP1A2CYP2C9PKM
SCHEMBL14366360 0.92 LTA4H (0.48) LMNAGAACYP1A2CYP2C9PKM
SCHEMBL25325632 0.86 LMNA (0.48) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL1453272 0.85 CA4 (0.48) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL11210416 0.84 LMNA (0.47) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL1252991 0.82 LMNA (0.45) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL10764289 0.82 LMNA (0.45) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL19714108 0.82 LMNA (0.45) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL17892009 0.82 LMNA (0.45) LMNAMTNR1AMTNR1BGAACYP1A2
SCHEMBL17901028 0.82 LMNA (0.45) LMNAMTNR1AMTNR1BGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230094112-A1 METHODS TO CONTROL INFECTION USING NEW GENERATION SMALL MOLECULE GROWTH INHIBITORS OHIO STATE INNOVATION FOUNDATION 2023-03-30 US disclosed
US-11478454-B2 Methods to control infection using new generation small molecule growth inhibitors OHIO STATE INNOVATION FOUNDATION (US) 2022-10-25 US disclosed
US-20200405691-A1 METHODS TO CONTROL INFECTION USING NEW GENERATION SMALL MOLECULE GROWTH INHIBITORS OHIO STATE INNOVATION FOUNDATION 2020-12-31 US disclosed
US-20110184418-A1 Unsealed, Non-Colloidal Radiopharmaceutical Compositions and Methods for Treatment of Abnormal Tissue SARI ASHER, LLC 2011-07-28 US disclosed
WO-2011035024-A2 UNSEALED, NON-COLLOIDAL RADIOPHARMACEUTICAL COMPOSITIONS AND METHODS FOR TREATMENT OF ABNORMAL TISSUE SARI ASHER LLC (US) 2011-03-24 WO disclosed
EP-1315517-B1 MIMETIC PEPTIDES FOR EPITOPE OF APOLIPOPROTEIN B-100, CONCATEMER AND MODIFIED PEPTIDES THEREOF, AND THE VACCINE COMPOSITION COMPRISING THE SAME KIM HYO JOON (KR) 2010-10-20 EP disclosed
US-20080138728-A1 LATENT ELECTROSTATIC IMAGE BEARING MEMBER, AND IMAGE FORMING APPARATUS, IMAGE FORMING METHOD AND PROCESS CARTRIDGE USING THE SAME RICOH COMPANY, LTD. (JP) 2008-06-12 US disclosed
US-20060025390-A1 Treatment of hormone allergy and related symptoms and disorders ROBY RUSSELL R 2006-02-02 US disclosed
WO-2005105106-A2 HORMONE TREATMENT OF MACULAR DEGENERATION ROBY RUSSELL R (US) 2005-11-10 WO disclosed
WO-2005105107-A2 HORMONE TREATMENT OF MULTIPLE SCLEROSIS ROBY RUSSELL R (US) 2005-11-10 WO disclosed
US-20050239757-A1 Hormone treatment of macular degeneration ROBY RUSSELL R 2005-10-27 US disclosed
US-20050239758-A1 Hormone treatment of multiple sclerosis ROBY RUSSELL R 2005-10-27 US disclosed
EP-1315517-A4 MIMETIC PEPTIDES FOR EPITOPE OF APOLIPOPROTEIN B-100, CONCATEMER AND MODIFIED PEPTIDES THEREOF, AND THE VACCINE COMPOSITION COMPRISING THE SAME KIM HYO JOON (KR) 2005-02-09 EP disclosed
US-6825318-B2 VACCINE FOR OBESITY THERAPY; HYBRID POLYPEPTIDES Kim, Hyo-Joon (KR) 2004-11-30 US disclosed
US-20030211997-A1 Mimetic peptides for an epitope of apolipoprotein B-100, concatemers of the peptides, and modified peptides, and compositions comprising the same KIM, HYO-JOON (KR) 2003-11-13 US disclosed
EP-1315517-A1 MIMETIC PEPTIDES FOR EPITOPE OF APOLIPOPROTEIN B-100, CONCATEMER AND MODIFIED PEPTIDES THEREOF, AND THE VACCINE COMPOSITION COMPRISING THE SAME Kim, Hyo-Joon (KR) 2003-06-04 EP disclosed
WO-2003024468-A1 SUBSTANCES EXTRACTED FROM CORN WHICH CAN INHIBIT THE ACTIVITIES OF AMYLASE, PHARMACEUTICAL COMPOSITIONS AND FOOD ADDITIVES CONTAINING THE SAME EXTRACTS FOR TREATMENT OR PREVENTION OF OBESITY AND DIABETES MELLITUS, AND PROCESSES FOR THEIR PREPARATIONS BIONEER CORPORATION (KR) 2003-03-27 WO disclosed
WO-2002020040-A1 MIMETIC PEPTIDES FOR EPITOPE OF APOLIPOPROTEIN B-100, CONCATEMER AND MODIFIED PEPTIDES THEREOF, AND THE VACCINE COMPOSITION COMPRISING THE SAME KIM HYO JOON (KR) 2002-03-14 WO disclosed
WO-1993011669-A1 USE OF 3-PHENYLURACIL DERIVATIVES FOR THE DESICCATION AND ABSCISSION OF PLANT PARTS BASF AKTIENGESELLSCHAFT (DE) 1993-06-24 WO disclosed
US-4388081-A CONTAINING PHENOXYALCOHOL AS ANTINKNOCK ADDITIVE PHILLIPS PETROLEUM COMPANY (US) 1983-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11478454-B2 Methods to control infection using new generation small molecule growth inhibitors SMURF1, SMURF2, SMYD3 LMNA 4633/4885MTNR1A 3180/4885MTNR1B 3199/4885
US-20230094112-A1 METHODS TO CONTROL INFECTION USING NEW GENERATION SMALL MOLECULE GROWTH INHIBITORS SMURF1, SMURF2, SMYD3 LMNA 4604/4885MTNR1A 3213/4885MTNR1B 3201/4885
US-20200405691-A1 METHODS TO CONTROL INFECTION USING NEW GENERATION SMALL MOLECULE GROWTH INHIBITORS SMURF1, SMURF2, SMYD3 LMNA 4633/4885MTNR1A 3180/4885MTNR1B 3199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.