SCHEMBL14965508

SCHEMBL14965508

N#Cc1ccc(-c2cc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)ccn2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 1/20 0.37
SRC P12931 1/20 0.36
TBK1 Q9UHD2 2/20 0.35
CYP11B1 P15538 1/20 0.35
KCNH2 Q12809 2/20 0.34
KCNJ1 P48048 1/20 0.34
TGFBR1 P36897 2/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
IKBKE Q14164 1/20 0.33
COMT P21964 1/20 0.33
MOK Q9UQ07 1/20 0.33
USP30 Q70CQ3 1/20 0.33
LRRK2 Q5S007 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965986 0.88 KCNJ1 (0.41) CYP11B1KCNH2KCNJ1MAPTSMN1; SMN2
SCHEMBL14966215 0.87 CYP11B1 (0.43) CAMKK2SRCCYP11B1KCNH2KCNJ1
SCHEMBL14966317 0.86 LOXL2 (0.42) TGFBR1HTR1ADRD2SMN1; SMN2MAPKAPK2
SCHEMBL14966162 0.86 CHRM1 (0.36) KCNH2TGFBR1HTR1ADRD2SMN1; SMN2
SCHEMBL14965795 0.86 CYP11B1 (0.45) SRCCYP11B1KCNH2KCNJ1HTR1A
SCHEMBL14965790 0.84 DRD2 (0.38) SRCCYP11B1KCNH2KCNJ1HTR1A
SCHEMBL14965683 0.83 DRD2 (0.43) KCNH2HTR1ADRD2
SCHEMBL14965893 0.83 SCN9A (0.37) SRCCYP11B1KCNH2KCNJ1HTR1A
SCHEMBL14965635 0.82 ALDH1A1 (0.42) KCNH2KCNJ1MAPTSMN1; SMN2
SCHEMBL14966336 0.82 DRD2 (0.45) CYP11B1KCNH2KCNJ1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed