SCHEMBL14965795

SCHEMBL14965795

N#Cc1ccc(-c2cccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.45
CHRM3 P20309 2/20 0.40
DRD2 P14416 5/20 0.39
HTR1A P08908 3/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
DRD4 P21917 2/20 0.37
DRD3 P35462 2/20 0.37
SLC2A1 P11166 2/20 0.37
KDM1A O60341 1/20 0.36
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
MCHR1 Q99705 1/20 0.36
NMT1 P30419 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966336 0.94 DRD2 (0.45) CYP11B1CHRM3DRD2HTR1AROCK2
SCHEMBL14965764 0.91 MCHR1 (0.42) DRD2HTR1AROCK2ROCK1SLC2A1
SCHEMBL14965986 0.91 KCNJ1 (0.41) CYP11B1KCNJ1KCNH2
SCHEMBL14971091 0.90 DRD2 (0.44) DRD2HTR1ADRD4DRD3MCHR1
SCHEMBL14965790 0.89 DRD2 (0.38) CYP11B1DRD2HTR1ADRD4DRD3
SCHEMBL14966205 0.87 LSS (0.46) DRD2HTR1AROCK2ROCK1DRD4
SCHEMBL14965508 0.86 CAMKK2 (0.37) CYP11B1DRD2HTR1ASRCKCNJ1
SCHEMBL14966131 0.85 DRD2 (0.49) CHRM3DRD2HTR1ADRD4DRD3
SCHEMBL14965893 0.84 SCN9A (0.37) CYP11B1DRD2HTR1ASLC2A1SRC
SCHEMBL14966240 0.84 KIT (0.40) CYP11B1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed