SCHEMBL14965690

SCHEMBL14965690

CN1CCN(C(=O)c2ccc(-c3ccc(CN4CCOc5nc([N+](=O)[O-])cn5CC4)cc3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.54
CHKA P35790 2/20 0.54
LSS P48449 2/20 0.45
PKM P14618 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
GALR3 O60755 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 4/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 1/20 0.42
BLM P54132 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HPGD P15428 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965840 0.97 HRH3 (0.57) HRH3CHKAPKMNPSR1SMN1; SMN2
SCHEMBL14965949 0.92 HPGD (0.51) HRH3CHKALSSPKMNPSR1
SCHEMBL14965684 0.92 CHKA (0.45) HRH3CHKASMN1; SMN2ALDH1A1MEN1
SCHEMBL14965948 0.91 HPGD (0.50) HRH3CHKALSSPKMNPSR1
SCHEMBL14966002 0.89 HPGD (0.54) HRH3CHKAPKMNPSR1SMN1; SMN2
SCHEMBL14965793 0.88 HPGD (0.53) HRH3PKMNPSR1SMN1; SMN2KDM4E
SCHEMBL14965941 0.88 HRH3 (0.46) HRH3LSSPKMNPSR1SMN1; SMN2
SCHEMBL14965877 0.88 MET (0.42) HRH3CHKASMN1; SMN2ALDH1A1HTT
SCHEMBL14965368 0.86 KCNJ1 (0.40) HRH3LSSPKMNPSR1SMN1; SMN2
SCHEMBL14971065 0.86 SLC2A1 (0.41) HRH3PKMNPSR1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed