SCHEMBL14965877

SCHEMBL14965877

CN1CCN(C(=O)c2ccc(-c3ccc(CN4CCOc5nc([N+](=O)[O-])cn5CC4)cc3)cc2F)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.42
CHKA P35790 2/20 0.41
HRH3 Q9Y5N1 1/20 0.40
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MELK Q14680 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966081 0.92 KCNJ1 (0.39) ALDH1A1POLBLMNAHTTSMN1; SMN2
SCHEMBL14966238 0.91 MET (0.41) METHRH3LMNAHTTSMN1; SMN2
SCHEMBL14965806 0.90 MET (0.39) METLMNAHTTSMN1; SMN2JAK2
SCHEMBL14965690 0.88 HRH3 (0.54) CHKAHRH3ALDH1A1POLBHTT
SCHEMBL14966153 0.88 JAK2 (0.38) METALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL14965684 0.87 CHKA (0.45) CHKAHRH3ALDH1A1LMNAHTT
SCHEMBL14965662 0.87 ALDH1A1 (0.38) ALDH1A1POLBLMNAHTTSMN1; SMN2
SCHEMBL14966035 0.87 MCHR1 (0.42) METALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL14966144 0.85 JAK2 (0.38) METHRH3LMNAHTTSMN1; SMN2
SCHEMBL14965840 0.85 HRH3 (0.57) CHKAHRH3ALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed