SCHEMBL14965756

SCHEMBL14965756

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)NC1CC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
ALDH1A1 P00352 5/20 0.37
AHR P35869 1/20 0.37
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
OGA O60502 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966168 0.96 ALDH1A1 (0.40) ALDH1A1POLBKDM4ELMNAHPGD
SCHEMBL14965807 0.88 SIGMAR1 (0.52) SMN1; SMN2SIGMAR1
SCHEMBL14965832 0.86 NPC1 (0.36) PKMALDH1A1AHRPOLBLMNA
SCHEMBL14966113 0.84 POLB (0.39) PKMALDH1A1AHRPOLBSMN1; SMN2
SCHEMBL14965582 0.83 HSD17B10 (0.38) ALDH1A1AHRPOLBLMNAL3MBTL1
SCHEMBL14969489 0.83 ALDH1A1 (0.43) ALDH1A1AHRPOLBKDM4ESMN1; SMN2
SCHEMBL14966161 0.83 NPC1 (0.42) ALDH1A1AHRPOLBKDM4ELMNA
SCHEMBL14965902 0.82 KDM4E (0.53) ALDH1A1KDM4ESMN1; SMN2SIGMAR1
SCHEMBL14966018 0.81 POLB (0.49) ALDH1A1AHRPOLBKDM4ELMNA
SCHEMBL14965889 0.80 ALDH1A1 (0.44) PKMALDH1A1POLBKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed