SCHEMBL14965902

SCHEMBL14965902

O=C(NC1CC1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
KMT2A Q03164 3/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
DRD4 P21917 1/20 0.49
TMEM97 Q5BJF2 4/20 0.48
MCHR1 Q99705 3/20 0.45
ALDH1A1 P00352 3/20 0.43
FGFR1 P11362 1/20 0.43
FGFR2 P21802 1/20 0.43
FGFR3 P22607 1/20 0.43
MEN1 O00255 2/20 0.43
SIGMAR1 Q99720 2/20 0.42
SLC6A12 P48065 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966188 0.97 KDM4E (0.50) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14966181 0.96 KDM4E (0.56) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14965672 0.89 DRD4 (0.47) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14965796 0.88 MCHR1 (0.45) KDM4EKMT2AMCHR1ALDH1A1MEN1
SCHEMBL14965370 0.86 ALDH1A1 (0.44) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14965407 0.86 KCNJ1 (0.42) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14969456 0.85 POLB (0.43) KDM4EKMT2ASMN1; SMN2MCHR1ALDH1A1
SCHEMBL14965822 0.85 FGFR1 (0.45) KDM4EDRD4MCHR1FGFR1FGFR2
SCHEMBL14965322 0.85 KMT2A (0.45) KDM4EKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL14965777 0.85 HIF1A (0.58) KDM4EKMT2ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed