SCHEMBL14965764

SCHEMBL14965764

N#Cc1cccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 9/20 0.42
SLC2A1 P11166 1/20 0.42
TNIK Q9UKE5 1/20 0.40
PRKAA2 P54646 1/20 0.40
KCNJ1 P48048 1/20 0.40
KCNH2 Q12809 1/20 0.40
MET P08581 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966336 0.94 DRD2 (0.45) MCHR1SLC2A1TNIKKCNJ1KCNH2
SCHEMBL14965795 0.91 CYP11B1 (0.45) MCHR1SLC2A1KCNJ1KCNH2HTR1A
SCHEMBL14965986 0.91 KCNJ1 (0.41) PRKAA2KCNJ1KCNH2
SCHEMBL14971108 0.87 ALDH1A1 (0.44) KCNJ1
SCHEMBL14965746 0.86 DRD2 (0.41) SLC2A1KCNJ1KCNH2DRD2
SCHEMBL14971091 0.84 DRD2 (0.44) MCHR1HTR1ADRD2
SCHEMBL14965511 0.84 LTA4H (0.40) SLC2A1
SCHEMBL14966132 0.84 DRD4 (0.44) MCHR1SLC2A1HTR1ADRD2ADORA2A
SCHEMBL14965626 0.84 LTA4H (0.40) SLC2A1
SCHEMBL14965761 0.84 S1PR5 (0.44) KCNJ1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed