SCHEMBL14965822

SCHEMBL14965822

O=C(NC1CC1)c1cc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.45
FGFR2 P21802 1/20 0.45
FGFR3 P22607 1/20 0.45
CNR1 P21554 3/20 0.40
CNR2 P34972 3/20 0.40
CCR3 P51677 1/20 0.40
DRD4 P21917 1/20 0.39
PDE4B Q07343 2/20 0.38
PRKAA2 P54646 1/20 0.38
MCHR1 Q99705 4/20 0.38
USP30 Q70CQ3 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965650 0.97 CNR1 (0.42) FGFR1FGFR2FGFR3CNR1CNR2
SCHEMBL14966145 0.91 FGFR1 (0.43) FGFR1FGFR2FGFR3CCR3DRD4
SCHEMBL14965563 0.91 MCHR1 (0.42) FGFR1FGFR2FGFR3CNR1CNR2
SCHEMBL14965814 0.89 FGFR1 (0.41) FGFR1FGFR2FGFR3CNR1CNR2
SCHEMBL14966019 0.88 MCHR1 (0.39) MCHR1
SCHEMBL14966188 0.88 KDM4E (0.50) FGFR1FGFR2FGFR3CCR3DRD4
SCHEMBL14965848 0.88 MCHR1 (0.37) MCHR1
SCHEMBL14966086 0.88 FGFR1 (0.38) FGFR1FGFR2FGFR3CNR1CNR2
SCHEMBL14965672 0.87 DRD4 (0.47) CCR3DRD4MCHR1KDM4E
SCHEMBL14965509 0.85 FGFR1 (0.42) FGFR1FGFR2FGFR3CCR3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed