SCHEMBL14966019

SCHEMBL14966019

CCNC(=O)c1cc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.39
HSP90AA1 P07900 11/20 0.38
HSP90AB1 P08238 11/20 0.38
MTOR P42345 1/20 0.37
KCNH2 Q12809 1/20 0.37
SLC2A1 P11166 1/20 0.36
DHODH Q02127 1/20 0.35
CHRM4 P08173 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965970 0.91 MTOR (0.39) MCHR1HSP90AA1HSP90AB1MTORKCNH2
SCHEMBL14965848 0.90 MCHR1 (0.37) MCHR1KCNH2SLC2A1DHODH
SCHEMBL14965822 0.88 FGFR1 (0.45) MCHR1
SCHEMBL14966204 0.88 SLC2A1 (0.42) MCHR1HSP90AA1HSP90AB1SLC2A1
SCHEMBL14965956 0.87 MTOR (0.39) HSP90AA1HSP90AB1MTORKCNH2SLC2A1
SCHEMBL14965650 0.87 CNR1 (0.42) MCHR1HSP90AA1
SCHEMBL14965896 0.87 SUCNR1 (0.40) MCHR1HSP90AA1HSP90AB1SLC2A1
SCHEMBL14965662 0.86 ALDH1A1 (0.38) MCHR1
SCHEMBL14966035 0.86 MCHR1 (0.42) MCHR1KCNH2CHRM4
SCHEMBL14965597 0.85 MTOR (0.39) MCHR1HSP90AA1HSP90AB1MTORKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed