SCHEMBL14965672

SCHEMBL14965672

O=C(NC1CC1)c1cccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.47
TMEM97 Q5BJF2 2/20 0.47
DRD2 P14416 1/20 0.47
ALDH1A1 P00352 1/20 0.44
MCHR1 Q99705 3/20 0.43
SMO Q99835 1/20 0.43
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CCR3 P51677 1/20 0.41
MAPK14 Q16539 1/20 0.41
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966188 0.92 KDM4E (0.50) DRD4TMEM97DRD2ALDH1A1MCHR1
SCHEMBL14965511 0.89 LTA4H (0.40) ALDH1A1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL14965626 0.89 LTA4H (0.40) ALDH1A1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL14965902 0.89 KDM4E (0.53) DRD4TMEM97ALDH1A1MCHR1KDM4E
SCHEMBL14965896 0.88 SUCNR1 (0.40) ALDH1A1MCHR1KMT2AMEN1
SCHEMBL14969471 0.88 KDM4E (0.41) ALDH1A1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL14965822 0.87 FGFR1 (0.45) DRD4MCHR1KDM4ECCR3
SCHEMBL14966181 0.86 KDM4E (0.56) DRD4TMEM97ALDH1A1MCHR1KDM4E
SCHEMBL14966243 0.85 TNIK (0.45) DRD2ALDH1A1KMT2AMEN1ACHE
SCHEMBL14965650 0.84 CNR1 (0.42) DRD4MCHR1KDM4EKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed