SCHEMBL14965844

SCHEMBL14965844

O=C(c1cc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cn2)ccc1F)N1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
STAT3 P40763 4/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
PARP1 P09874 1/20 0.34
ATR Q13535 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
HTR2C P28335 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965820 0.94 JAK2 (0.37) LMNAHTTSTAT3MEN1KMT2A
SCHEMBL14966144 0.94 JAK2 (0.38) LMNAHTTSTAT3JAK2JAK1
SCHEMBL14965662 0.91 ALDH1A1 (0.38) LMNAHTTALDH1A1POLBPARP1
SCHEMBL14965678 0.88 MTOR (0.37) MCHR1
SCHEMBL14966238 0.88 MET (0.41) LMNAHTTSTAT3JAK2JAK1
SCHEMBL14966157 0.88 AVPR1B (0.38) HTR2CMCHR1
SCHEMBL14965805 0.87 DHODH (0.36) STAT3JAK2JAK1TYK2JAK3
SCHEMBL14965970 0.87 MTOR (0.39) HTR2CMCHR1
SCHEMBL14965814 0.87 FGFR1 (0.41) KMT2AALDH1A1SMN1; SMN2MCHR1
SCHEMBL14966145 0.86 FGFR1 (0.43) JAK2JAK1TYK2JAK3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed