SCHEMBL14965820

SCHEMBL14965820

O=C(c1ccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cn2)cc1F)N1CCCC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.37
JAK1 P23458 2/20 0.37
TYK2 P29597 2/20 0.37
JAK3 P52333 2/20 0.37
STAT3 P40763 4/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MTOR P42345 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
MET P08581 1/20 0.34
PIK3CA P42336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965844 0.94 LMNA (0.35) JAK2JAK1TYK2JAK3STAT3
SCHEMBL14966238 0.94 MET (0.41) JAK2JAK1TYK2JAK3STAT3
SCHEMBL14965805 0.92 DHODH (0.36) JAK2JAK1TYK2JAK3STAT3
SCHEMBL14965835 0.90 MTOR (0.37) JAK2JAK1TYK2JAK3LMNA
SCHEMBL14965652 0.88 GPR119 (0.38) JAK2JAK1TYK2JAK3MET
SCHEMBL14965830 0.88 AVPR1B (0.36) MET
SCHEMBL14966144 0.88 JAK2 (0.38) JAK2JAK1TYK2JAK3STAT3
SCHEMBL14965597 0.87 MTOR (0.39) MTORMET
SCHEMBL14965487 0.87 FGFR1 (0.39) MET
SCHEMBL14965509 0.86 FGFR1 (0.42) MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed