SCHEMBL14965947

SCHEMBL14965947

CC(C)(C)[Si](C)(C)OCCN(CCn1cc([N+](=O)[O-])nc1[N+](=O)[O-])Cc1cccc(OC(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 1/20 0.37
MITF O75030 1/20 0.34
PPARA Q07869 4/20 0.33
PPARD Q03181 3/20 0.33
ALKBH1 Q13686 1/20 0.32
NR1D1 P20393 1/20 0.31
NR1H3 Q13133 1/20 0.31
PPARG P37231 3/20 0.31
TLR7 Q9NYK1 3/20 0.31
SLC6A9 P48067 3/20 0.31
CYP2D6 P10635 2/20 0.31
CYP3A4 P08684 1/20 0.31
LMNA P02545 1/20 0.30
KCNH2 Q12809 2/20 0.30
SLC6A5 Q9Y345 1/20 0.30
P2RX7 Q99572 1/20 0.30
GRK2 P25098 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966156 0.91 KCNH2 (0.37) SLC6A9CYP2D6CYP3A4KCNH2SLC6A5
SCHEMBL14965763 0.90 MITF (0.34) MITFLMNAKCNH2
SCHEMBL14965539 0.87 NR1H3 (0.39) MITFNR1D1NR1H3
SCHEMBL14965901 0.86 MITF (0.37) MITFCYP2D6LMNA
SCHEMBL14971075 0.84 MEP1B (0.38) MEP1BMITFPPARAPPARDALKBH1
SCHEMBL14965734 0.83 NR1D1 (0.38) MITFNR1D1NR1H3LMNA
SCHEMBL14969412 0.82 NR1D1 (0.36) MITFNR1D1NR1H3KCNH2
SCHEMBL14966100 0.82 KCNH2 (0.40) MITFKCNH2
SCHEMBL14969684 0.82 NR1D1 (0.36) MITFNR1D1LMNA
SCHEMBL14965850 0.79 MITF (0.35) MITFLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed