SCHEMBL14966100

SCHEMBL14966100

CC(C)(C)[Si](C)(C)OCCN(CCn1cc([N+](=O)[O-])nc1[N+](=O)[O-])Cc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.40
CHRM1 P11229 1/20 0.39
MITF O75030 1/20 0.34
SLC6A4 P31645 3/20 0.33
PTGS1 P23219 1/20 0.33
SLC6A2 P23975 1/20 0.33
TXNRD1 Q16881 1/20 0.33
SOS1 Q07889 1/20 0.32
TRPM8 Q7Z2W7 2/20 0.32
SLC6A3 Q01959 2/20 0.32
TRPA1 O75762 1/20 0.31
ALDH1A1 P00352 1/20 0.30
OPRM1 P35372 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966156 0.91 KCNH2 (0.37) KCNH2
SCHEMBL14969412 0.91 NR1D1 (0.36) KCNH2MITFSOS1ALDH1A1OPRM1
SCHEMBL14965763 0.90 MITF (0.34) KCNH2MITFSOS1TRPA1OPRM1
SCHEMBL14969684 0.90 NR1D1 (0.36) MITFSOS1ALDH1A1
SCHEMBL14965901 0.88 MITF (0.37) MITFSOS1ALDH1A1
SCHEMBL14965539 0.83 NR1H3 (0.39) MITFALDH1A1
SCHEMBL14971142 0.83 KCNH2 (0.39) KCNH2CHRM1MITFSLC6A4PTGS1
SCHEMBL14965734 0.82 NR1D1 (0.38) MITFALDH1A1
SCHEMBL14965947 0.82 MEP1B (0.37) KCNH2MITF
SCHEMBL14965850 0.80 MITF (0.35) MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed