SCHEMBL14965896

SCHEMBL14965896

CCNC(=O)c1cccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 1/20 0.40
ALDH1A1 P00352 4/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
CHRM3 P20309 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HSP90AA1 P07900 2/20 0.39
HSP90AB1 P08238 2/20 0.39
MCHR1 Q99705 1/20 0.38
TNIK Q9UKE5 1/20 0.38
SLC2A1 P11166 1/20 0.38
WNT1 P04628 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966204 0.92 SLC2A1 (0.42) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL14969471 0.90 KDM4E (0.41) SUCNR1ALDH1A1LMNAMAPTMEN1
SCHEMBL14965370 0.89 ALDH1A1 (0.44) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL14965626 0.88 LTA4H (0.40) SUCNR1ALDH1A1LMNAMAPTMEN1
SCHEMBL14965511 0.88 LTA4H (0.40) SUCNR1ALDH1A1LMNAMAPTMEN1
SCHEMBL14965672 0.88 DRD4 (0.47) ALDH1A1MEN1KMT2AMCHR1
SCHEMBL14971109 0.87 TP53 (0.40) ALDH1A1LMNAMAPTSLC2A1
SCHEMBL14966243 0.87 TNIK (0.45) SUCNR1ALDH1A1LMNAMAPTMEN1
SCHEMBL14966019 0.87 MCHR1 (0.39) HSP90AA1HSP90AB1MCHR1SLC2A1
SCHEMBL14965684 0.85 CHKA (0.45) SUCNR1ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed