SCHEMBL14966151

SCHEMBL14966151

O=C(NCc1ccc(C(F)(F)F)cc1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1.O=C(NCc1ccc(OC(F)F)cc1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1.O=C(NCc1cccc(OC(F)F)c1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.42
ALDH1A1 P00352 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
TSHR P16473 1/20 0.40
GLS O94925 1/20 0.39
MAPK14 Q16539 3/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ROCK2 O75116 3/20 0.38
ROCK1 Q13464 2/20 0.38
HIF1A Q16665 2/20 0.38
EPAS1 Q99814 2/20 0.38
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966210 0.94 ALDH1A1 (0.43) ALDH1A1HDAC4HDAC6TSHRROCK2
SCHEMBL14965754 0.91 TSHR (0.47) ALDH1A1HDAC4HDAC6TSHRMAPT
SCHEMBL14965591 0.89 CHRM3 (0.47) CHRM3ALDH1A1HDAC4HDAC6TSHR
SCHEMBL14965538 0.88 HDAC4 (0.49) CHRM3ALDH1A1HDAC4HDAC6TSHR
SCHEMBL14966045 0.86 TSHR (0.50) CHRM3ALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL14965737 0.84 CHRM1 (0.49) ALDH1A1HDAC4HDAC6TSHR
SCHEMBL14965927 0.83 ALDH1A1 (0.52) ALDH1A1TSHRMAPTSMN1; SMN2HIF1A
SCHEMBL14965722 0.83 KLKB1 (0.48) CHRM3ALDH1A1HDAC4HDAC6TSHR
SCHEMBL14965800 0.83 ALDH1A1 (0.58) ALDH1A1HDAC4HDAC6TSHRSMN1; SMN2
SCHEMBL14966118 0.83 ALDH1A1 (0.39) ALDH1A1MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed