SCHEMBL14966152

SCHEMBL14966152

O=C(Nc1cccc(OC(F)(F)F)c1)c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
RAB9A P51151 5/20 0.50
NPC1 O15118 4/20 0.50
TP53 P04637 2/20 0.50
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ABL1 P00519 1/20 0.48
KCNH2 Q12809 1/20 0.48
CHRM1 P11229 1/20 0.45
MAPT P10636 3/20 0.44
KDM4E B2RXH2 2/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.44
HIF1A Q16665 3/20 0.44
EPAS1 Q99814 3/20 0.44
TNF P01375 1/20 0.42
NOD2 Q9HC29 1/20 0.42
NOD1 Q9Y239 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965916 0.93 ABL1 (0.56) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14965787 0.92 HIF1A (0.44) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14965927 0.92 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14966147 0.91 KCNH2 (0.53) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14965959 0.91 KCNH2 (0.53) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14969414 0.90 LMNA (0.53) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14965591 0.89 CHRM3 (0.47) ALDH1A1KMT2AMEN1ABL1KCNH2
SCHEMBL14966245 0.89 MEN1 (0.53) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL14965884 0.88 CHRM1 (0.46) ALDH1A1KMT2AMEN1ABL1KCNH2
SCHEMBL14965557 0.86 DRD4 (0.48) ALDH1A1KMT2AMEN1KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed