SCHEMBL14966207

SCHEMBL14966207

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(NCc3ccc(OC(F)F)cc3)n1)CC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.37
IDH1 O75874 6/20 0.36
OGA O60502 3/20 0.36
KCNH2 Q12809 4/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
HRH4 Q9H3N8 5/20 0.34
HRH3 Q9Y5N1 3/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
SLC6A2 P23975 2/20 0.33
HTR1D P28221 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
HRH2 P25021 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
HTR5A P47898 1/20 0.33
HTR6 P50406 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965573 0.89 CHRM1 (0.50) CHRM1IDH1OGAKCNH2CCNC
SCHEMBL14965834 0.87 OGA (0.49) IDH1OGAHRH4HRH3ADRA2B
SCHEMBL14965593 0.86 MET (0.39) CHRM1OGAKCNH2HRH4HRH3
SCHEMBL14966122 0.81 OGA (0.41) IDH1OGAHRH4HRH3ADRA2B
SCHEMBL14965871 0.80 ALDH1A1 (0.42) OGAHTR6
SCHEMBL14965841 0.80 OGA (0.46) CHRM1OGAHRH4HRH3ADRA2B
SCHEMBL14965923 0.78 OGA (0.46) OGAKCNH2HRH4HRH3ADRA2B
SCHEMBL14965636 0.78 HRH4 (0.47) IDH1OGAHRH4HRH3ADRA2B
SCHEMBL14966015 0.78 CHRM1 (0.44) CHRM1KCNH2
SCHEMBL14965804 0.76 KMT2A (0.41) CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed