SCHEMBL14965636

SCHEMBL14965636

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(NCC3CCCCC3)n1)CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 9/20 0.47
IDH1 O75874 1/20 0.45
CXCR4 P61073 1/20 0.38
OGA O60502 5/20 0.37
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
SLC6A2 P23975 2/20 0.36
HTR1D P28221 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HRH3 Q9Y5N1 3/20 0.34
CDC7 O00311 2/20 0.34
ROCK2 O75116 1/20 0.34
CCNB2 O95067 1/20 0.34
MAP4K4 O95819 1/20 0.34
CDK1 P06493 1/20 0.34
RET P07949 1/20 0.34
CCNB1 P14635 1/20 0.34
PRKACA P17612 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965834 0.83 OGA (0.49) HRH4IDH1OGAADRA2BADRA2C
SCHEMBL14965871 0.82 ALDH1A1 (0.42) OGAALDH1A1HTR6
SCHEMBL14965593 0.80 MET (0.39) HRH4OGAADRA2BADRA2CSLC6A2
SCHEMBL14966122 0.79 OGA (0.41) HRH4IDH1OGAADRA2BADRA2C
SCHEMBL14965841 0.78 OGA (0.46) HRH4OGAADRA2BADRA2CSLC6A2
SCHEMBL14965923 0.78 OGA (0.46) HRH4OGAADRA2BADRA2CSLC6A2
SCHEMBL14965573 0.78 CHRM1 (0.50) HRH4IDH1OGASLC6A2HRH3
SCHEMBL14966207 0.78 CHRM1 (0.37) HRH4IDH1OGAADRA2BADRA2C
SCHEMBL14965943 0.78 GBA1 (0.40) ALDH1A1
SCHEMBL14965617 0.77 TRPV1 (0.45) OGAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed