SCHEMBL14965834

SCHEMBL14965834

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(NCc3ccccc3)n1)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGA O60502 4/20 0.49
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
SLC6A2 P23975 1/20 0.45
HRH2 P25021 1/20 0.45
HTR1D P28221 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR7 P34969 1/20 0.45
HTR2B P41595 1/20 0.45
HTR5A P47898 1/20 0.45
HTR6 P50406 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
IDH1 O75874 5/20 0.43
PIK3CB P42338 4/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966122 0.90 OGA (0.41) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965593 0.89 MET (0.39) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965871 0.88 ALDH1A1 (0.42) OGAHTR6PKMMAPTALDH1A1
SCHEMBL14966207 0.87 CHRM1 (0.37) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965573 0.87 CHRM1 (0.50) OGASLC6A2HRH4HRH3IDH1
SCHEMBL14965636 0.83 HRH4 (0.47) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965923 0.82 OGA (0.46) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965841 0.82 OGA (0.46) OGAADRA2BADRA2CSLC6A2HRH2
SCHEMBL14965984 0.80 MAPT (0.42) ACHEMAPTALDH1A1TDP1L3MBTL1
SCHEMBL14965617 0.80 TRPV1 (0.45) OGAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed